Search on: PENTAZOCINE 
Descriptors Found: 1
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Descriptor English:   Pentazocine 
Descriptor Spanish:   Pentazocina 
Descriptor Portuguese:   Pentazocina 
Synonyms English:   Fortral
Hydrochloride, Pentazocine
Lactate, Pentazocine
Lexir
Pentazocine Hydrochloride
Pentazocine Lactate
Talwin  
Tree Number:   D03.132.577.249.106.700
D04.615.723.795.106.700
Definition English:   The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor. (From AMA Drug Evaluations Annual, 1991, p97) 
Pharmacological Action:   Analgesics, Opioid
Adjuvants, Anesthesia
Narcotic Antagonists
Narcotics
 
History Note English:   66(64) 
Allowable Qualifiers English:  
AD administration & dosage AE adverse effects
AG agonists AA analogs & derivatives
AN analysis AI antagonists & inhibitors
BL blood CF cerebrospinal fluid
CS chemical synthesis CH chemistry
CL classification EC economics
HI history IM immunology
IP isolation & purification ME metabolism
PK pharmacokinetics PD pharmacology
PO poisoning RE radiation effects
ST standards SD supply & distribution
TU therapeutic use TO toxicity
UR urine  
Record Number:   10617 
Unique Identifier:   D010423 

Occurrence in VHL:
 

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