Expresión de búsqueda:
MFN=57545
Descriptores Encontrados:
1
Mostrando:
1 .. 1
1 / 1
DeCS
Descriptor
Inglés
:
Sunitinib
Descriptor
Español
:
Sunitinib
Descriptor
Portugués
:
Sunitinibe
Sinónimos
Inglés
:
5-(5-Fluoro-2-oxo-1,2-dihydroindolylidenemethyl)-2,4-dimethyl-1H-pyrrole-3-carboxylic acid (2-diethylaminoethyl)amide
SU 011248
SU 11248
SU-011248
SU-11248
SU011248
SU11248
Sunitinib Malate
Sutent
Categoría:
D03.383.129.578.823
D03.633.100.473.877
Definición
Inglés
:
An indole and pyrrole derivative that inhibits VEGFR-2 and PDGFR BETA RECEPTOR
TYROSINE
KINASES. It is used as an antineoplastic agent for the treatment of
GASTROINTESTINAL STROMAL TUMORS
, and for treatment of advanced or metastatic RENAL CELL
CARCINOMA.
Acción Farmacológica:
Antineoplastic Agents
Angiogenesis Inhibitors
Protein Kinase Inhibitors
Nota Histórica
Inglés
:
2019 (2003)
Calificadores Permitidos
Inglés
:
AD
administration & dosage
AE
adverse effects
AG
agonists
AA
analogs & derivatives
AN
analysis
AI
antagonists & inhibitors
BL
blood
CF
cerebrospinal fluid
CS
chemical synthesis
CH
chemistry
CL
classification
EC
economics
HI
history
IM
immunology
IP
isolation & purification
ME
metabolism
PK
pharmacokinetics
PD
pharmacology
PO
poisoning
RE
radiation effects
ST
standards
SD
supply & distribution
TU
therapeutic use
TO
toxicity
UR
urine
Número del Registro:
57545
Identificador Único:
D000077210
Ocurrencia en la BVS
:
Similar:
DeCS